Acylation of lycoctonine: semi-synthesis of inuline, delsemine analogues and methyllycaconitine
1994
Blagbrough, I.S. | Coates, P.A. | Hardick, D.J. | Lewis, T. | Rowan, M.G. | Wonnacott, S. | Potter, B.V.L.
Lycoctonine has been acylated to afford sequentially inuline, delsemine analogues and methyllycaconitine using isatoic anhydride followed by S-(-)-methylsuccinic anhydride. This protocol is a rapid, facile method for the regiospecific introduction of the anthranilate ester moiety found in potent nicotinic acetylcholine receptor antagonists.
Show more [+] Less [-]AGROVOC Keywords
Bibliographic information
This bibliographic record has been provided by National Agricultural Library