C–H Bond Functionalization of Tetrahydropyridopyrimidines and Other Related Hetereocycles
2017
Cheng, Zhanling | Yu, Zhiliang | Yang, Song | Shen, Hong C. | Zhao, Weili | Zhong, Sheng
A novel and efficient 2-step method for the functionalization of the C–H bond adjacent to the amino group of tetrahydropyridopyrimidine (THPP) is reported herein. The reaction features mild conditions and excellent tolerance of a wide range of functional groups. Moreover, this method is applicable to tetrahydroisoquinolone (THIQ), which provides a useful supplement to literature method. This method gives chemists a new tool to functionalize a C–H bond at late stage and may find applications in both synthetic organic and medicinal chemistry.
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