Stereoselective synthesis of tetrahydro-2H-[2]benzopyrano[3,4-c]pyrrol-3-ones and related compounds as precursors of serotonin 5-HT₂C receptor agonists
2011
Francis, Stuart | Kiyoi, Takao | Reid, Mark | Davies, Keneth | Laats, Steven | M'Arthur, Duncan | Feilden, Helen | Easson, Anna Marie | Kiyoi, Yasuko | Wishart, Grant | Ray, Peter
Tetrahydro-2H-[2]benzopyrano[3,4-c]pyrrol-3-ones and the related 3a-methyl-2,3,3a,4,5,9b-hexahydro-1H-benzo[e]isoindole analogues were synthesised by an intramolecular Diels–Alder reaction. The observed stereoselectivity was dependent upon the nature of the tethered dienophile as well as the judicious placement of the amide.
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