Pd-catalyzed Suzuki/Sonogashira cross-coupling reaction and the direct sp3 arylation of 7-chloro-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidine
2018
Loubidi, Mohammed | Moutardier, Anaïs | Campos, Joana F. | Berteina-Raboin, Sabine
A rapid and efficient method is reported for the synthesis of the [1,2,4]triazolo[1,5-a]pyrimidine motif. Palladium catalyzed Suzuki and Sonogashira cross coupling reactions on 7-chloro-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidine were performed. The direct sp3 arylation of compounds resulting from the Suzuki reaction was then carried out.
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书目信息
出版者
Elsevier B.V.
其它主题
Suzuki reaction; Suzuki; 5-a]pyrimidine; Triazolo[1; Sonogashira; Direct sp3 arylation; Arylation
语言
英语
类型
Journal Article; Text
2024-02-28
MODS