Arginine thioacid in synthesis of arginine conjugates and peptides

Khaybullin, Ravil N.; Panda, Siva S.; Mirzai, Saeid; Toneff, Ellen; Asiri, Abdullah M.; Hall, C Dennis; Katritzky, Alan R.

Arginine thioacid in synthesis of arginine conjugates and peptides

2014

Protected arginine thioacid enables convenient N-acylation with no detectable racemization. We report efficient syntheses of potentially biologically active arginine conjugates and novel arginine-containing di-, tri- and tetrapeptides in good yields without loss of chiral integrity.

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