Regioselectivity of Larock Indole Synthesis Using Functionalized Alkynes
2008
SUGINO, Kumi | YOSHIMURA, Hiroshi | NISHIKAWA, Toshio | Isobe, Minoru
Regioselectivity of Larock indole synthesis, a palladium-catalyzed heteroannulation between o-iodoaniline and internal acetylene, was estimated using acetylenes substituted with ester and/or Boc-protected amine at the homopropargylic position and with perbenzyl- and unprotected glucose. Low to moderate regioselectivities were observed in all the cases, indicating these functional groups do not exert good directing effects, in the Larock indole synthesis.
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书目信息
出版者
Japan Society for Bioscience, Biotechnology, and Agrochemistry
其它主题
Regioselectivity; Larock indole synthesis
语言
英语
注释
Nal-ap-2-clean
类型
Journal Article; Text
2024-02-28
2026-02-03
MODS